Custom Peptides
Cayman Chemical RheIn-8-glucosIde 10mg
An anthraquinone glycoside; increases the rate of sennoside A metabolism by mouse intestinal bacteria in vitro at 0.03-1 mM; increases the purgative activity of sennoside A in mice in a dose-dependent manner; inhibits PTP1B (IC50 = 11.5 μM); metabolized to rhein by intestinal bacteria
Cayman Chemical 6-MAPBhydrochlorIde 10mg
An analytical reference standard categorized as a benzofuran; intended for research and forensic applications
Cayman Chemical PropylhexedrInhydrochLRId 10mg
An α-adrenergic sympathomimetic amine that acts as a local vasoconstrictor; intended for research and forensic applications
Cayman Chemical OlIgomycIn B 10mg
A nonselective inhibitor of the mitochondrial F1FO ATP synthase that can reduce the rate of ATP depletion in myocardial ischemia and decrease calcium-induced calcium release oscillation frequency of rat sensory neurons
Cayman Chemical BromosporIn 10mg
A non-selective bromodomain inhibitor that at 1 µM has been shown to accelerate FRAP recovery of BRD4 and CREBBP bromodomains in HeLa cells
Cayman Chemical 7Methoxy8 3morpholIn4yl 10mg
A building block; has been used in the synthesis of PI3K inhibitors
Cayman Chemical SLP7111228hydrochlorIde 10mg
A potent and selective SPHK1 inhibitor (Kis = 0.048 and >10 μM for SPHK1 and 2, respectively); induces a concentration-dependent decrease in U937 cells; decreases blood levels of S1P in a dose-dependent manner in rats
Cayman Chemical PncuronIumbromIde hydrate 10mg
An antagonist of muscle-type nAChRs (IC50 = 14.8 nM); acts as a non-depolarizing neuromuscular blocking agent; enhances isoflurane anesthesia (ED50 = 1.62 UG/kg to reduce immobilization)
Cayman Chemical EIcosapentaenoyl ChlorIde 10mg
A derivative of eicosapentaenoic acid; has been used in the synthesis of fatty acid conjugates to enhance lipophilicity and cell permeability of bioactive compounds
Cayman Chemical Boc-Glu-OBzl 1g
An amino acid building block; has been used in the synthesis of peptide-based inhibitors of human caspases and HRV 3C protease that have enzyme inhibitory activity in vitro
Cayman Chemical NpTosylGlyProLyspNAac 10mg
A colorimetric plasmin substrate; hydrolysis releases pNA, which can be quantified by colorimetric detection at 405 nm as a measure of plasmin activity